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Amphetamine is understood to inhibit monoamine oxidase, whereas the flexibility of amphetamine and its metabolites to inhibit many P450 isozymes and also other enzymes has not been sufficiently elucidated. In vitro experiments with human microsomes show minor inhibition of CYP2D6 by amphetamine and insignificant inhibition of CYP1A2, 2D6, and 3A4 b